Multi‐Drug‐Resistance‐Reverting Agents: 2‐Aryloxazole and 2‐Arylthiazole Derivatives as Potent BCRP or MRP1 Inhibitors
2009 · ChemMedChem · 51 citations
https://doi.org/10.1002/cmdc.200800329
M
Marialessandra Contino
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Marialessandra Contino is an academic researcher from University of Bari Aldo Moro. The author has contributed to research in topics: Pharmacological Receptor Mechanisms and Effects & Drug Transport and Resistance Mechanisms & Receptor Mechanisms and Signaling. The author has an h-index of 34, co-authored 119 publications.
ORCID: 0000-0002-0713-3151Papers by this author
worksSAR Studies on Tetrahydroisoquinoline Derivatives: The Role of Flexibility and Bioisosterism To Raise Potency and Selectivity toward P-glycoprotein
2014 · Journal of Medicinal Chemistry · 31 citations
https://doi.org/10.1021/jm501640e
Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug resistance (MDR) modulators
2019 · European Journal of Medicinal Chemistry · 28 citations
https://doi.org/10.1016/j.ejmech.2019.03.054
Naphthalenyl derivatives for hitting P-gp/MRP1/BCRP transporters
2012 · Bioorganic & Medicinal Chemistry · 27 citations
https://doi.org/10.1016/j.bmc.2012.12.021
The interaction of celecoxib with MDR transporters enhances the activity of mitomycin C in a bladder cancer cell line
2013 · Molecular Cancer · 16 citations
https://doi.org/10.1186/1476-4598-12-47
A Benzopyrane Derivative as a P‐Glycoprotein Stimulator: A Potential Agent to Decrease β‐Amyloid Accumulation in Alzheimer’s Disease
2011 · ChemMedChem · 14 citations
https://doi.org/10.1002/cmdc.201100469
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